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PFI-1
CAS No. 1403764-72-6
PFI-1 ( PF-6405761 )
Catalog No. M11688 CAS No. 1403764-72-6
PFI-1 is a selective BET (bromodomain-containing protein) inhibitor for BRD4 with IC50 of 0.22 μM in a cell-free assay.
Purity : >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 39 | In Stock |
|
| 10MG | 63 | In Stock |
|
| 25MG | 111 | In Stock |
|
| 50MG | 178 | In Stock |
|
| 100MG | 327 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NamePFI-1
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NoteResearch use only, not for human use.
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Brief DescriptionPFI-1 is a selective BET (bromodomain-containing protein) inhibitor for BRD4 with IC50 of 0.22 μM in a cell-free assay.
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DescriptionPFI-1 is a selective BET (bromodomain-containing protein) inhibitor for BRD4 with IC50 of 0.22 μM in a cell-free assay.
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SynonymsPF-6405761
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PathwayChromatin/Epigenetic
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TargetEpigenetic Reader Domain
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RecptorBRD2; BRD4
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number1403764-72-6
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Formula Weight347.39
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Molecular FormulaC16H17N3O4S
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Purity>98%(HPLC)
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SolubilityDMSO: 69 mg/mL (198.62 mM)
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SMILESO=S(C1=CC=CC=C1OC)(NC2=CC3=C(NC(N(C)C3)=O)C=C2)=O
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Chemical Name2-methoxy-N-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-6-yl)benzenesulfonamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Fish PV, et al. J Med Chem, 2012, 55(22), 9831-9837.
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